Kinase Inhibitors to Watch

Kinase Inhibitors Archive Kinases are extremely important enzymes that control much of how the cells in our body function. Mutations, deletions or mangling of the structure of a regulatory kinase can play havoc with the particular protein and the cell function it is supposed to control. Most if not all human cancers are thought to be caused by one or more malfunctioning kinases. PCI-32765 and CAL-101 are two targeted, designer-made oral drugs currently in clinical trials.